BDBM271020 7-(benzenesulfonyl)-4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-methyl-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 138

SMILES Cc1nc(N2C[C@@H](C)O[C@@H](C)C2)c2[nH]c(N)c(S(=O)(=O)c3ccccc3)c2n1

InChI Key InChIKey=XMYWVTITRZCPIM-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 271020   

TargetFree fatty acid receptor 2(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 271020BDBM271020(7-(benzenesulfonyl)-4-[(2R,6S)-2,6-dimethylmorphol...)
Affinity DataEC50:  6nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
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Date in BDB:
12/11/2018
Entry Details
US Patent