BDBM271146 7-(3-fluorobenzenesulfonyl)-4-(2-methylmorpholin-4-yl)-2-(trifluoromethyl)-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 265

SMILES CC1CN(CCO1)c1nc(nc2c(c(N)[nH]c12)S(=O)(=O)c1cccc(F)c1)C(F)(F)F

InChI Key InChIKey=ZCLXTKTUOWMZDZ-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 271146   

TargetFree fatty acid receptor 2(Human)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM271146(7-(3-fluorobenzenesulfonyl)-4-(2-methylmorpholin-4...)
Affinity DataEC50:  3nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
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Date in BDB:
12/11/2018
Entry Details
US Patent