BDBM272800 (S)-2-((1-(2- aminobenzo[d]oxazol- 5-yl)-8,9-dihydro- 7H-6-oxa-2,9a- diazabenzo[cd]azulen-4- yl)amino)propanamide::US10065970, Compound 105::US10435414, Compound 105
SMILES C[C@H](Nc1cc2OCCCn3c(nc(c1)c23)-c1ccc2oc(N)nc2c1)C(N)=O
InChI Key InChIKey=IQKZEIMSEKFAGN-JTQLQIEISA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 272800
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Genentech
US Patent
Genentech
US Patent
Affinity DataKi: 0.0320nMAssay Description:PI3K Binding assays are intended for determining the biochemical potency of small molecule PI3K inhibitors. The PI3K lipid kinase reaction is perform...More data for this Ligand-Target Pair