BDBM279804 PMPeG, prodrug::US10035814, Compound 142820

SMILES C=C(COCP(=O)(OCOC(=O)OC(C)C)OCOC(=O)OC(C)C)Cn1cnc2c(=O)[nH]c(N)nc21

InChI Key InChIKey=UIRRNQBNTZJDSC-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 279804   

TargetTelomerase protein component 1(Human)
Geron

US Patent
LigandChemical structure of BindingDB Monomer ID 279804BDBM279804(US10035814, Compound 142820 | PMPeG, prodrug)
Affinity DataEC50:  1.09E+4nMAssay Description:Telomerase inhibition is observed in cells following the addition of the prodrugs (R)-PMPG-diisopropyloxy ester or (S)-PMPG-diisopropyloxy ester. HT3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2018
Entry Details
US Patent