BDBM293974 (2S)-4-((4-(5-((4-(1-(1H- Tetrazol-5-yl)pent-3-yn-2- yl)phenoxy)methyl)benzo[b] thiophen-3-yl)-3- methylphenoxy)methyl)-4- hydroxytetrahydro-2H- thiopyran 1,1-dioxide::US10106553, Compound 6

SMILES CC#C[C@@H](Cc1nnn[nH]1)c1ccc(OCc2ccc3sc(Cl)c(-c4ccc(OCC5(O)CCS(=O)(=O)CC5)cc4C)c3c2)cc1

InChI Key

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 293974   

TargetFree fatty acid receptor 1(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM293974((2S)-4-((4-(5-((4-(1-(1H- Tetrazol-5-yl)pent-3-yn-...)
Affinity DataEC50:  190nMT: 25°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent