BDBM293974 (2S)-4-((4-(5-((4-(1-(1H- Tetrazol-5-yl)pent-3-yn-2- yl)phenoxy)methyl)benzo[b] thiophen-3-yl)-3- methylphenoxy)methyl)-4- hydroxytetrahydro-2H- thiopyran 1,1-dioxide::US10106553, Compound 6
SMILES CC#C[C@@H](Cc1nnn[nH]1)c1ccc(OCc2ccc3sc(Cl)c(-c4ccc(OCC5(O)CCS(=O)(=O)CC5)cc4C)c3c2)cc1
InChI Key
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 293974
Affinity DataEC50: 190nMT: 25°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair