BDBM297845 5-[5-Oxo-7-(piperidin-4-yl)-4,5-dihydropyrazolo[1,5-a]pyrimidin-3-yl]thiophene-3-carbonitrile trifluoroacetate::US10118930, Example 68

SMILES N#Cc1csc(-c2cnn3c(C4CCNCC4)cc(=O)[nH]c23)c1

InChI Key InChIKey=QTJGEGYBQOVETK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 297845   

TargetTissue-type plasminogen activator(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandChemical structure of BindingDB Monomer ID 297845BDBM297845(US10118930, Example 68 | 5-[5-Oxo-7-(piperidin-4-y...)
Affinity DataIC50: 11nMAssay Description:The clot-lysis test system configures the kinetics of clot formation and degradation in vitro and allows quantifying modulation of the process by sel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent