BDBM298055 3-[4-(2-fluorophenyl)-1,3-thiazol-2-yl]-7-(piperidin-4-yl)pyrazolo[1,5-c]pyrimidin-5(4H)-one hydrochloride::US10118930, Example 267

SMILES O=c1cc(C2CCNCC2)n2ncc(-c3nc(-c4ccccc4F)cs3)c2[nH]1

InChI Key InChIKey=GSDBCUXSOHRFLB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 298055   

TargetTissue-type plasminogen activator(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandChemical structure of BindingDB Monomer ID 298055BDBM298055(US10118930, Example 267 | 3-[4-(2-fluorophenyl)-1,...)
Affinity DataIC50: 15nMAssay Description:The clot-lysis test system configures the kinetics of clot formation and degradation in vitro and allows quantifying modulation of the process by sel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent