BDBM298114 3-[(3,3-difluoroazetidin-1-yl)carbonyl]-7-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidin-5 (4H)-one hydrochloride::US10118930, Example 326

SMILES O=C(c1cnn2c(C3CCNCC3)cc(=O)[nH]c12)N1CC(F)(F)C1

InChI Key InChIKey=JHXIJHNLAHUGCP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 298114   

TargetTissue-type plasminogen activator(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandChemical structure of BindingDB Monomer ID 298114BDBM298114(US10118930, Example 326 | 3-[(3,3-difluoroazetidin...)
Affinity DataIC50: 12nMAssay Description:The clot-lysis test system configures the kinetics of clot formation and degradation in vitro and allows quantifying modulation of the process by sel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent