BDBM304033 5,8-Dimethyl-2-(2-phenyl-1H-benzimidazol-5-yl)[1,2,4]triazolo[1,5-a]pyrazine::US10138245, Example 4

SMILES Cc1ncc(C)n2nc(-c3ccc4[nH]c(-c5ccccc5)nc4c3)nc12

InChI Key InChIKey=ZOZHIFOCCJPYGJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 304033   

LigandChemical structure of BindingDB Monomer ID 304033BDBM304033(5,8-Dimethyl-2-(2-phenyl-1H-benzimidazol-5-yl)[1,2...)
Affinity DataIC50: 27nMAssay Description:Recombinant human phosphodiesterase 10A (PDE10A) purified to homogeneity from Sf9 cells overexpressing PDE10A gene (GenBank/EMBL accession number: NM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent