BDBM31638 tetrahydrobenzothiophene (THBT), 13a

SMILES CC(C)(C)C1CCc2c(C1)sc(NC(=O)c1c(F)cccc1F)c2C(N)=O

InChI Key InChIKey=ORUPXWFIFZMHMP-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 31638   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Gsk

LigandBDBM31638(tetrahydrobenzothiophene (THBT), 13a)Copy SMILESCopy InChI

Affinity DataIC50:  79nMpH: 7.5 T: 23°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair

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