BDBM3254 (1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5-dihydroxy-4-({2-hydroxy-6-[(propan-2-yloxy)carbonyl]phenyl}carbonyl)benzoate::Balanol Benzophenone Ester Analog 9

SMILES CC(C)OC(=O)c1cccc(O)c1C(=O)c1c(O)cc(cc1O)C(=O)O[C@@H]1CCC[C@H]1NC(=O)c1ccc(O)cc1

InChI Key InChIKey=XDTAJQIDTGQFQG-HYBUGGRVSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 3254   

TargetProtein kinase C alpha type(Homo sapiens (Human))
Sphinx Pharmaceuticals

LigandPNGBDBM3254((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50:  4.70E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
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TargetProtein kinase C beta type(Homo sapiens (Human))
Sphinx Pharmaceuticals

LigandPNGBDBM3254((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50:  440nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
Sphinx Pharmaceuticals

LigandPNGBDBM3254((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50:  260nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Sphinx Pharmaceuticals

LigandPNGBDBM3254((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50:  1.30E+4nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C delta type(Homo sapiens (Human))
Sphinx Pharmaceuticals

LigandPNGBDBM3254((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50:  50nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails Article