BDBM336817 (S)-4-((6-(1,2-dihydroxyethyl)- 2-(4-(4-(trifluoromethoxy)- phenoxy)phenyl)pyrimidin-4- yl)methyl)piperazin-2-one::US9745287, Compound 41
SMILES OC[C@@H](O)c1cc(CN2CCNC(=O)C2)nc(n1)-c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1
InChI Key InChIKey=HTZGXLVJGBQQPM-OAQYLSRUSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 336817
Affinity DataKi: 875nMAssay Description:Cells Manual Electrophysiology: The hNav1.7 expressing HEK-293 cells are plated on 35 mm culture dishes pre-coated with poly-D-lysine in standard DME...More data for this Ligand-Target Pair
Affinity DataIC50: 1.19E+3nMAssay Description:Assay Buffer: The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL...More data for this Ligand-Target Pair