BDBM346441 US10202378, Example 54::isobutyl 4-[(3R)-3-hydroxy-3-(5-methylisoxazol-3-yl)but-1-ynyl]-6-methyl-7-oxo-1H-pyrrolo[2,3-c]pyridine-3-carboxylate
SMILES CC(C)COC(=O)c1c[nH]c2c1c(cn(C)c2=O)C#C[C@@](C)(O)c1cc(C)on1
InChI Key
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 346441
TargetTranscription initiation factor TFIID subunit 1 [1381-1497](Homo sapiens (human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 179nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1 [1504-1635](Homo sapiens (Human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 122nMAssay Description:His/Flag epitope tagged TAF1-BD21504-1635 was cloned, expressed, and purified to homogeneity. TAF1-BD2 binding and inhibition was assessed by monitor...More data for this Ligand-Target Pair