BDBM35666 BMC173130 Compound 1t::benzazepinelidene acetamide derivative, 1b
SMILES Cc1ccn(n1)-c1ccc(C(=O)N2CCC(F)(F)\C(=C/C(=O)NCCO)c3ccccc23)c(Cl)c1
InChI Key InChIKey=XKZZIPLEGIRBDK-HKWRFOASSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 35666
Affinity DataKi: 9.70nM ΔG°: -10.9kcal/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
Affinity DataKi: 9.70nM ΔG°: -10.9kcal/molepH: 7.4 T: 23°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
Affinity DataKi: 28nM ΔG°: -10.3kcal/moleT: 25°CAssay Description:Chinese hamster ovary (CHO) cells stably expressing human V1a receptors. Cells were washed with phosphate buffered saline, and then collected in ice-...More data for this Ligand-Target Pair
Affinity DataKi: 28nM ΔG°: -10.2kcal/molepH: 7.4 T: 23°CAssay Description:Chinese hamster ovary (CHO) cells stably expressing human V1a receptors. Cells were washed with phosphate buffered saline, and then collected in ice-...More data for this Ligand-Target Pair