BDBM35710 benzazepine derivative, 17

SMILES CN(C)C1CCCN(C(=O)c2ccc(NC(=O)c3ccccc3C)cc2)c2cccc(Cl)c12

InChI Key InChIKey=OGPADXVSAFOLGB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 35710   

TargetVasopressin V1a receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35710(benzazepine derivative, 17)
Affinity DataIC50:  1.70E+3nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35710(benzazepine derivative, 17)
Affinity DataIC50:  190nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed