BDBM369506 N,2-dimethyl-N-[2-[4-[[(R, 2S)-2-phenylcyclopropyl]amino]-1-piperidyl]ethyl]pyridin-4-amine::US10233152, Example 44

SMILES CN(CCN1CCC(CC1)N[C@@H]1C[C@H]1c1ccccc1)c1ccnc(C)c1

InChI Key InChIKey=RWEBWBGUJGIGHO-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 369506   

TargetLysine-specific histone demethylase 1A(Human)
Mirati Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 369506BDBM369506(N,2-dimethyl-N-[2-[4-[[(R, 2S)-2-phenylcyclopropyl...)
Affinity DataIC50: 9nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent