BDBM373553 1-((4-Cyclopropanemethylamino)-6-(2,6-dimethylphenoxy)-7-fluoroquinazolin-2-yl)-1H-pyrazole-4-carboxylic acid;::US10246442, Example 15::US10975062, Example 15
SMILES Cc1cccc(C)c1Oc1cc2c(NCC3CC3)nc(nc2cc1F)-n1cc(cn1)C(O)=O
InChI Key InChIKey=XFUJIDZIIMBAQL-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 373553
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair