BDBM3753 N-(3-bromophenyl)-9H-pyrimido[4,5-b]indol-4-amine::Pyrimido[4,5-b]indole deriv. 44

SMILES Brc1cccc(Nc2ncnc3[nH]c4ccccc4c23)c1

InChI Key InChIKey=MHRKNNUUCCNFPI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 3753   

TargetEpidermal growth factor receptor(Human)
Parke-Davis Pharmaceutical Research

LigandPNGBDBM3753(N-(3-bromophenyl)-9H-pyrimido[4,5-b]indol-4-amine ...)
Affinity DataIC50: 31nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2005
Entry Details Article
PubMed