BDBM387067 1-(4-Methoxyphenyl)-7-oxo-6-(3-(3-oxomorpholino)-3-azabicyclo[3.1.0]hexan-6-yl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide::US9938272, Example 13

SMILES COc1ccc(cc1)-n1nc(C(N)=O)c2CCN(C3C4CN(CC34)N3CCOCC3=O)C(=O)c12

InChI Key InChIKey=BJRVNAXOOOCMPW-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 387067   

TargetCoagulation factor X(Human)
North China Pharmaceutical

US Patent
LigandPNGBDBM387067(1-(4-Methoxyphenyl)-7-oxo-6-(3-(3-oxomorpholino)-3...)
Affinity DataKi:  30nMAssay Description:Factor Xa (human or rat): In the assay for measuring the inhibition of human or rat factor Xa activity, Tris-HCl buffer (50 mM, pH 8.3, 150 mM NaCl) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent