BDBM391686 3-{[4-({[(1R,2S)-2-phenylcyclopropyl]amino}methyl)-1-(pyridin-2-ylmethyl)piperidin-4-yl]methyl}benzoic Acid::US10300051, Example 32
SMILES OC(=O)c1cccc(CC2(CN[C@@H]3CC3c3ccccc3)CCN(Cc3ccccn3)CC2)c1
InChI Key InChIKey=IYWXJGBPAAKFCT-SSYAZFEXSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 391686
Affinity DataIC50: <100nMAssay Description:LANCE LSD1/KDM1A demethylase assay—10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair