BDBM401751 US10005792, Compound 110

SMILES COc1ccc(CN(C[C@H](O)CNC(=O)c2ccnc(NC3CN(C3)C(C)=O)c2)C2Cc3ccccc3C2)c(OC)c1

InChI Key InChIKey=XBOMTZOKLUWLBP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 401751   

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401751(US10005792, Compound 110)
Affinity DataIC50: 166nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent