BDBM405637 US10351547, Compound 2-55::US10597377, Compound 2-55

SMILES CCCNCC1CN(c2c(-c3cc(C)cc(F)c3)cnc3ccc(-c4cc(F)c5[nH]c(=O)[nH]c5c4)cc23)C1

InChI Key InChIKey=KTJPCMIVPPTHDM-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 405637   

TargetSomatostatin receptor type 2(Human)
Crinetics Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 405637BDBM405637(US10351547, Compound 2-55 | US10597377, Compound 2...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
US Patent

TargetSomatostatin receptor type 2(Human)
Crinetics Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 405637BDBM405637(US10351547, Compound 2-55 | US10597377, Compound 2...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC # CCL-61) stably expressing the human SSTR2 are plated in each well of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent