BDBM405748 US10351547, Compound 2-218

SMILES CO[C@@H]1CN(CC[C@H]1N)c1c(cnc2ccc(cc12)-c1cccc(C#N)c1NC(=O)OC)-c1cc(C)cc(F)c1

InChI Key InChIKey=DMRJPEQGTGMFOH-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 405748   

TargetSomatostatin receptor type 2(Human)
Crinetics Pharmaceuticals

US Patent
LigandPNGBDBM405748(US10351547, Compound 2-218)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
US Patent