BDBM412455 N-(5-(2-cyclopropoxy-5-(1-methyl- 1H-pyrazol-4-yl)phenyl)pyrazin-2- yl)-4-methylnicotinamide::US10399967, Compound 86

SMILES Cc1ccncc1C(=O)Nc1cnc(cn1)-c1cc(ccc1OC1CC1)-c1cnn(C)c1

InChI Key InChIKey=QWVKAZFNEIYDFE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412455   

TargetInterleukin-2(Human)
Prcl Research

US Patent
LigandChemical structure of BindingDB Monomer ID 412455BDBM412455(US10399967, Compound 86 | N-(5-(2-cyclopropoxy-5-(...)
Affinity DataIC50: 61nMAssay Description:Human peripheral blood mononuclear cells (PBMCs) are prepared from heparinized human blood by separation over a Ficoll density gradient.PBMCs are sti...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
US Patent