BDBM413128 (R)-4-(1-(5-(4-ethyl-3-methylpiperazine-1-carbonyl)pyridin-2-yl)-5-hydroxy-1H-pyrazol-4-yl)-2-fluoro-5-methylbenzonitrile::US10407409, Example 395
SMILES CCN1CCN(C[C@H]1C)C(=O)c1ccc(nc1)-n1ncc(c1O)-c1cc(F)c(cc1C)C#N
InChI Key InChIKey=KAOROSNDUNJDEV-MRXNPFEDSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 413128
Affinity DataIC50: 3.31nMAssay Description:The IC50 values for the PHD2 enzyme (residues 181-417) were determined by mixing increasing amounts of inhibitor with a fixed amount of enzyme (5 nM,...More data for this Ligand-Target Pair
Ligand Info