BDBM420059 N-(azetidin-2-ylmethyl)-2-cyclopentyl-10-methyl- 1-oxo-1,2-dihydropyrazino[1,2-a]indole-4- carboxamide::US10487087, Compound 22

SMILES Cc1c2ccccc2n2c(cn(C3CCCC3)c(=O)c12)C(=O)NCC1CCN1

InChI Key InChIKey=YTHTWDLFQZVFEP-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 420059   

TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University

US Patent
LigandPNGBDBM420059(N-(azetidin-2-ylmethyl)-2-cyclopentyl-10-methyl- 1...)
Affinity DataEC50: >3.00E+4nMAssay Description:To assess the effects of test compounds on GLP-1 or glucagon potency and efficacy, a high-throughput calcium mobilization assay was used essentially ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/20/2020
Entry Details
US Patent