BDBM425903 US10512644, Compound Oxycodone

SMILES CN1CC[C@@]23[C@H]4Oc5c2c(CC1[C@]3(O)CC[C@@H]4O)ccc5CO

InChI Key

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 425903   

TargetMu-type opioid receptor(Human)
Inheris Pharmaceuticals

US Patent
LigandPNGBDBM425903(US10512644, Compound Oxycodone)
Affinity DataKi:  133nMAssay Description:Briefly, serial dilutions of the test compounds were placed in a 96-well plate to which were added SPA beads, membrane and radioligand. The assay con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Inheris Pharmaceuticals

US Patent
LigandPNGBDBM425903(US10512644, Compound Oxycodone)
Affinity DataEC50:  478nMAssay Description:Briefly, suspensions of cells expressing either the mu, kappa or delta opioid receptors were prepared in buffer containing 0.5 mM isobutyl-methyl xan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
US Patent