BDBM426138 5-[8-[4-(2-Fluoroethyl)-1-piperidyl]-2-phenyl-imidazo[1,2-a]pyrazin-3-::US10513523, Example 77
SMILES FCCC1CCN(CC1)c1nccn2c(c(nc12)-c1ccccc1)-c1ccc2NC(=O)Cc2c1
InChI Key InChIKey=IYGHATLDUFZHRF-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 426138
Affinity DataIC50: 0.400nMAssay Description:This assay was used to test compounds for their ability to inhibit TARP γ8 dependent AMPA receptor activity. The AMPA receptor is a non-selectiv...More data for this Ligand-Target Pair