BDBM437322 4-(benzyloxy)-1-methyl-5-(1-(1-phenylethyl)-1H- pyrazol-4-yl)pyridin-2(1H)-one::US10617680, Example 56::US11020380, Example 56

SMILES CC(c1ccccc1)n1cc(cn1)-c1cn(C)c(=O)cc1OCc1ccccc1

InChI Key InChIKey=XEKGESHSCFHZRB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437322   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437322(4-(benzyloxy)-1-methyl-5-(1-(1-phenylethyl)-1H- py...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437322(4-(benzyloxy)-1-methyl-5-(1-(1-phenylethyl)-1H- py...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent