BDBM437335 4-ethoxy-1-methyl-5-(1H-pyrazol-4-yl)pyridin-2(1H)-one::US10617680, Example 69::US11020380, Example 69

SMILES CCOc1cc(=O)n(C)cc1-c1cn[nH]c1

InChI Key InChIKey=XGDGIPOBQPRVHE-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437335   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437335(4-ethoxy-1-methyl-5-(1H-pyrazol-4-yl)pyridin-2(1H)...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437335(4-ethoxy-1-methyl-5-(1H-pyrazol-4-yl)pyridin-2(1H)...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent