BDBM437336 US10617680, Example 70::US11020380, Example 70::methyl-2-((4-(4-ethoxy-1-methyl-6-oxo-1,6-dihydropyridin- 3-yl)-1H-pyrazol-1-yl)methyl)benzoate

SMILES CCOc1cc(=O)n(C)cc1-c1cnn(Cc2ccccc2C(=O)OC)c1

InChI Key InChIKey=GMQFYLJWJJAYQU-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437336   

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM437336(methyl-2-((4-(4-ethoxy-1-methyl-6-oxo-1,6-dihydrop...)
Affinity DataIC50: 500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM437336(methyl-2-((4-(4-ethoxy-1-methyl-6-oxo-1,6-dihydrop...)
Affinity DataIC50: 500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2021
Entry Details
US Patent