BDBM437538 4-Methoxy-2-[4-(2'-methoxy-1-methyl-6-oxo-1,6-dihydro- [4,4']bipyridinyl-3-yl)-pyrazol-1-yl]-benzoic acid::US10617680, Example 272::US11020380, Example 272

SMILES COc1ccc(C(O)=O)c(c1)-n1cc(cn1)-c1cn(C)c(=O)cc1-c1ccnc(OC)c1

InChI Key InChIKey=RJJVHEFHDWJITN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437538   

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM437538(4-Methoxy-2-[4-(2'-methoxy-1-methyl-6-oxo-1,6-dihy...)
Affinity DataIC50: 500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2021
Entry Details
US Patent

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM437538(4-Methoxy-2-[4-(2'-methoxy-1-methyl-6-oxo-1,6-dihy...)
Affinity DataIC50: 500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent