BDBM438576 US10618902, Compound I-257

SMILES COc1cc(OC)c(Cl)c(c1Cl)-c1cc2cnc(Nc3cc(F)c(F)cc3NC(=O)C=C)nc2n(C)c1=O

InChI Key InChIKey=DLOLSKNBCRVLDG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 438576   

TargetFibroblast growth factor receptor 4(Human)
Celgene Car

US Patent
LigandPNGBDBM438576(US10618902, Compound I-257)
Affinity DataIC50: 500nMAssay Description:A 10× stock solution of FGFR4-WT (PR4380C or P3054), (from Invitrogen, Carlsbad, Calif.) corresponding to method a in Table 10, was prepared as descr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent