BDBM438592 US10618902, Compound I-273

SMILES CC(=O)N1CC(NC(=O)C=C)C(C1)Nc1ncc2cc(-c3cc(ccc3Cl)C(=O)Nc3cccc(c3)C(C)(C)C#N)c(=O)n(C)c2n1

InChI Key InChIKey=CBPAFKYINGPISM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 438592   

TargetFibroblast growth factor receptor 4(Human)
Celgene Car

US Patent
LigandPNGBDBM438592(US10618902, Compound I-273)
Affinity DataIC50: 500nMAssay Description:A 10× stock solution of FGFR4-WT (PR4380C or P3054), (from Invitrogen, Carlsbad, Calif.) corresponding to method a in Table 10, was prepared as descr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent