BDBM449015 US10696689, Compound 3-12

SMILES CNc1ncc(-c2cccc(F)c2)c(N2CCC3NCCOC3C2)c1-c1nc2c(OC)cc(cc2[nH]1)C#N

InChI Key InChIKey=FMTDRTIWTGCPLL-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 449015   

TargetSomatostatin receptor type 2(Human)
Crinetics Pharmaceuticals

US Patent
LigandPNGBDBM449015(US10696689, Compound 3-12)
Affinity DataEC50: >1nMAssay Description:On the day of the assay, the media is aspirated and the cells are treated with 50 μL of 1.6 μM NKH477 (Sigma # N3290) plus various dilution...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent