BDBM450715 US10676465, Example 91::US10676465, Example 92::ammonium 2-({4-[2-(5-chloropyridin-2- yl)-2-methyl-1,3-benzodioxol-4- yl]piperidin-1-yl}methyl)-1-(2- methoxyethyl)-1H-benzimidazole-6- carboxylate, ENT-X1 [from P8]
SMILES COCCn1c(CN2CCC(CC2)c2cccc3OC(C)(Oc23)c2ccc(Cl)cn2)nc2ccc(cc12)C([O-])=O
InChI Key InChIKey=QXJJCZYZPJIMDB-UHFFFAOYSA-M
Data 4 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 450715
Affinity DataEC50: 4.20nMAssay Description:GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de...More data for this Ligand-Target Pair
Affinity DataEC50: 72nMAssay Description:GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de...More data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de...More data for this Ligand-Target Pair