BDBM450722 US10676465, Example 98::US10676465, Example 99::ammonium 2-({4-[2-(4-cyano-2- fluorophenyl)-2-methyl-1,3-benzodioxol- 4-yl]piperidin-1-yl}methyl)-1-(1,3-oxazol- 2-ylmethyl)-1H-benzimidazole-6- carboxylate, ENT-X2 [from C83; footnote 12 in Table 2]
SMILES CC1(Oc2cccc(C3CCN(Cc4nc5ccc(cc5n4Cc4ncco4)C([O-])=O)CC3)c2O1)c1ccc(cc1F)C#N
InChI Key InChIKey=CVWLLOGSBBTZOM-UHFFFAOYSA-M
Data 4 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 450722
Affinity DataEC50: 2.80nMAssay Description:GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de...More data for this Ligand-Target Pair
Affinity DataEC50: 5.40nMAssay Description:GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de...More data for this Ligand-Target Pair
Affinity DataEC50: 440nMAssay Description:GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de...More data for this Ligand-Target Pair