BDBM47184 US8980905, 110::US9637499, Compound 110

SMILES FC(F)Oc1ccc(C(=O)Nc2c(Cl)cncc2Cl)c2OC3(CCSCC3)Oc12

InChI Key InChIKey=LXHMXTSEVTVMHJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 47184   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Leo Pharma

US Patent
LigandPNGBDBM47184(US8980905, 110 | US9637499, Compound 110)
Affinity DataIC50: 2nMAssay Description:Human recombinant PDE4 (Genbank accession no NM006203) was incubated for 1 hour, with the test compound at concentrations up to 10 μM, with cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2015
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Leo Pharma

US Patent
LigandPNGBDBM47184(US8980905, 110 | US9637499, Compound 110)
Affinity DataIC50: 2nMAssay Description:Human recombinant PDE4 (Genbank accession no NM_006203) was incubated for 1 hour, with the test compound at concentrations up to 10 μM, with cAM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2019
Entry Details
US Patent