BDBM471919 US10829446, Compound 154

SMILES Cc1cc(c(F)c(C(=O)NNS(=O)(=O)c2ccccc2)c1F)-c1ccccc1

InChI Key InChIKey=IEKZTZPMKNWIEF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 471919   

TargetHistone acetyltransferase KAT6A [507-778](Human)
Monash University

US Patent
LigandPNGBDBM471919(US10829446, Compound 154)
Affinity DataIC50: 10nMAssay Description:Active Moz protein was expressed as N-terminal fusion protein with a His6 tag in BL21 E. coli cells. Protein purification was performed via nickel-im...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent