BDBM47282 US9018217, Diisopropyl-(2-[2-[2-(5-methyl-[1,2,4]triazolo[1,5-a]pyridin-2-yl)-ethyl)-4-phenyl-imdazol-1-yl}-ethyl)-amine::US9592230, Diisopropyl-(2-[2-[2-(5-methyl-[1,2,4]triazolo[1,5-a]pyridin-2-yl)-ethyl]-4-phenyl-imidazol-1-yl}-ethyl)-amine

SMILES CC(C)N(CCn1cc(nc1CCc1nc2cccc(C)n2n1)-c1ccccc1)C(C)C

InChI Key InChIKey=SPAGVSXFBFHDCA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 47282   

LigandPNGBDBM47282(US9018217, Diisopropyl-(2-[2-[2-(5-methyl-[1,2,4]t...)
Affinity DataIC50: 7.30nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
US Patent

LigandPNGBDBM47282(US9018217, Diisopropyl-(2-[2-[2-(5-methyl-[1,2,4]t...)
Affinity DataIC50: 7.30nMAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2019
Entry Details
US Patent