BDBM481587 US10913710, Compound 5

SMILES CNc1ncc(Br)c(CN(CC2CCCCC2)S(=O)(=O)c2ccc(cc2)S(=O)(=O)N(CC2CCC(Cl)CC2)C2CCCC2)n1

InChI Key InChIKey=NIFYGKFNYNKRMN-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 481587   

TargetRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta(Human)
Max-Planck-Gesellschaft Zur Forderung Der Wissenschaften

US Patent
LigandPNGBDBM481587(US10913710, Compound 5)
Affinity DataKd:  65nMAssay Description:Binding to PDEδ was validated and quantified by means of a displacement assay employing a fluorescent-tagged analog of the HMG-CoA reductase inh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2021
Entry Details
US Patent