BDBM50002009 5-Chloro-1-(4-fluoro-phenyl)-3-piperidin-4-yl-1H-indole::CHEMBL273235

SMILES Fc1ccc(cc1)-n1cc(C2CCNCC2)c2cc(Cl)ccc12

InChI Key InChIKey=YCXCLZSLZGBCTA-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50002009   

TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002009(CHEMBL273235 | 5-Chloro-1-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002009(CHEMBL273235 | 5-Chloro-1-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 23nMAssay Description:Compound was tested for the inhibition of [3H]spiperone binding to dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50002009(CHEMBL273235 | 5-Chloro-1-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 204nMAssay Description:Inhibition of K+ channel activity in CHO cells expressing HERG Kv11.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50002009(CHEMBL273235 | 5-Chloro-1-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 204nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed