BDBM50011555 CHEMBL3262574::US9592235, Example 162::US9855269, Compound 5

SMILES Cc1cccc(c1)-c1ccc2ncnc(N)c2c1

InChI Key InChIKey=AOGXVQICAQYRPH-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50011555   

LigandPNGBDBM50011555(CHEMBL3262574 | US9592235, Example 162 | US9855269...)
Affinity DataIC50: 415nMAssay Description:The kinase activity of purified human MAP4K4 kinase domain was measured by monitoring the phosphorylation of a peptide substrate derived from moesin ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

LigandPNGBDBM50011555(CHEMBL3262574 | US9592235, Example 162 | US9855269...)
Affinity DataIC50: 415nMAssay Description:The kinase activity of purified human MAP4K4 kinase domain was measured by monitoring the phosphorylation of a peptide substrate derived from moesin ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2019
Entry Details
US Patent

LigandPNGBDBM50011555(CHEMBL3262574 | US9592235, Example 162 | US9855269...)
Affinity DataIC50: 423nMAssay Description:Inhibition of human MAP4K4 using 5-FAM-LGRDKYKTLRQIRQ-COOH as substrate by Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed