BDBM50015324 CHEMBL3264257

SMILES CN(C)CCNc1cncc(-c2ccc3[nH]cc(-c4ccnc(N)n4)c3c2)n1

InChI Key InChIKey=ILVKLFOUGPBUMK-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50015324   

TargetSerine/threonine-protein kinase pim-1(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015324BDBM50015324(CHEMBL3264257)
Affinity DataIC50: 3nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015324BDBM50015324(CHEMBL3264257)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of PIM1 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015324BDBM50015324(CHEMBL3264257)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of PIM3 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015324BDBM50015324(CHEMBL3264257)
Affinity DataIC50: 7nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015324BDBM50015324(CHEMBL3264257)
Affinity DataIC50: 110nMAssay Description:Inhibition of PIM2 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015324BDBM50015324(CHEMBL3264257)
Affinity DataIC50: 110nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed