BDBM50015325 CHEMBL3264258

SMILES CCN(CC)CCNc1cncc(-c2ccc3[nH]cc(-c4ccnc(N)n4)c3c2)n1

InChI Key InChIKey=UYOVRFLWHXLTBC-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50015325   

TargetSerine/threonine-protein kinase pim-1(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015325BDBM50015325(CHEMBL3264258)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of PIM1 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015325BDBM50015325(CHEMBL3264258)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of PIM3 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015325BDBM50015325(CHEMBL3264258)
Affinity DataIC50: 310nMAssay Description:Inhibition of PIM2 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed