BDBM50015328 CHEMBL3264261

SMILES CN(C)CCN(C)c1cncc(-c2ccc3[nH]cc(-c4ccnc(N)n4)c3c2)n1

InChI Key InChIKey=GAXARIICIJOJOY-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50015328   

TargetSerine/threonine-protein kinase pim-3(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015328BDBM50015328(CHEMBL3264261)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of PIM3 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015328BDBM50015328(CHEMBL3264261)
Affinity DataIC50: 8nMAssay Description:Inhibition of PIM1 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Keimyung University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015328BDBM50015328(CHEMBL3264261)
Affinity DataIC50: 180nMAssay Description:Inhibition of PIM2 kinase (unknown origin) using 5-FAM-labeled BAD peptide as substrate after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed