BDBM50017295 CHEMBL3288030

SMILES C[C@H]1CN(Cc2ccc(c(CN3CCOCC3)c2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)ccc3O)c2)C[C@@H](C)N1

InChI Key InChIKey=JHTLYFBBYQROBV-DZHYTCOUSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50017295   

LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human PDE4D using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50: >10nMAssay Description:Inhibition of human PDE4A1A using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50:  0.0251nMAssay Description:Inhibition of rat PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50017295(CHEMBL3288030)
Affinity DataIC50: >10nMAssay Description:Inhibition of human recombinant PDE4B at high-affinity rolipram binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed