BDBM50024284 CHEMBL3334979
SMILES COc1ccc(cc1OC)-c1cnc2scc(NC(=O)C3CCCCC3)c2c1
InChI Key InChIKey=HGVYGHNZFIZVJT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 24 hits for monomerid = 50024284
Affinity DataKd: 9nMAssay Description:Binding affinity to DRAK2 (unknown origin) ATP siteMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) using 33P-ATP after 30 mins by Trilux scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:Inhibition of DRAK2 (unknown origin) using 33P-ATP after 30 mins by Trilux scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Inhibition of DRAK1 (unknown origin) using 1 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Inhibition of DRAK1 (unknown origin) using 5 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 710nMAssay Description:Inhibition of DRAK1 (unknown origin) using 10 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:Inhibition of DRAK1 (unknown origin) using 25 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) using 50 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) using 100 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) using 250 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.91E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) using 500 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of DRAK2 (unknown origin) using 1 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of DRAK2 (unknown origin) using 5 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibition of DRAK2 (unknown origin) using 10 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of DRAK2 (unknown origin) using 25 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 720nMAssay Description:Inhibition of DRAK2 (unknown origin) using 50 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 990nMAssay Description:Inhibition of DRAK2 (unknown origin) using 100 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) using 250 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) using 500 uM ATP by biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
Affinity DataKd: 4.90nMAssay Description:Binding affinity to DRAK1 (unknown origin)More data for this Ligand-Target Pair