BDBM50032540 CHEMBL3354179

SMILES CCn1c(NC2CCCC2)nc2c(csc2c1=O)-c1cccnc1

InChI Key InChIKey=WYFACFDIJBGSEA-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50032540   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Kyoto 607-8042

Curated by ChEMBL
LigandPNGBDBM50032540(CHEMBL3354179)
Affinity DataIC50:  380nMAssay Description:Inhibition of human PDE4B1 expressed in insect cells assessed as inhibition of [3H]cAMP to [3H]AMP hydrolysis after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032540(CHEMBL3354179)
Affinity DataIC50:  2nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032540(CHEMBL3354179)
Affinity DataIC50:  2nMAssay Description:Inhibition of human PDE7A1 expressed in insect cells assessed as inhibition of [3H]cAMP to [3H]AMP hydrolysis after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed