BDBM50043290 CHEMBL3355038

SMILES COc1cc2ncnc(Nc3ccc4N(CCc4c3)C(=O)Cc3c(C)[nH]c4cc(F)ccc34)c2cc1OC

InChI Key InChIKey=NEWVPRAIGYZHJF-UHFFFAOYSA-N

Data  2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50043290   

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Dart Neuroscience

Curated by ChEMBL

LigandBDBM50043290(CHEMBL3355038)Copy SMILESCopy InChI

Affinity DataIC50: 0.631nMAssay Description:Inhibition of recombinant GST-tagged PERK (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
3/19/2016
Entry Details Article
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